WM-1119, KAT6A HAT inhibitor (TBI4013)
$108.00 – $351.00
KAT6A HAT inhibitor
SKU | Stock | SIZE (mg) | Price | Quantity | ||
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TBI4013-5MG | Yes | 5 MG | $108.00 | |||
TBI4013-25MG | Yes | 25 MG | $351.00 |
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Description
Product Details
Formal Name: 3-Fluoro-N’-(2-fluorophenyl)sulfonyl-5-pyridin-2-ylbenzohydrazide; 3-Fluoro-N’-(2-fluorobenzenesulfonyl)-5-(pyridine-2-yl)benzohydrazide
Molecular Formula: C18H13F2N3O3S
Formula Weight: 389.40
CAS Number: 2055397-28-7
Purity: >98%
Formulation: powder
Solubility: Soluble in DMSO (up to at least 25 mg/ml)
Storage: -20°C
Stability: ≥ 2 years.
Applications
KAT6A HAT inhibitor
Functions
Potent and selective inhibitor of the MYST family histone acetyltransferase KAT6A (MOZ) – IC50 = 6.3 nM. Induces cell cycle exit and cellular senescence without causing DNA damage. WM-1119 repressed the cell proliferation of sorafenib-resistant hepatocellular carcinoma cells.
Application Procedures
First dissolved in DMSO (up to at least 25 mg/ml), then diluted to aqueous buffer. Solutions in DMSO may be stored at -20°C for up to 3 months.
Additional information
SIZE (mg) | 25 MG, 5 MG |
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