SB-366791, TRPV1 blocker (TBI1217)

Description

Product Details

Formal Name: 3-(4-Chlorophenyl)-N-(3-methoxyphenyl)-2-propenamide

Molecular Formula: C₁₆H₁₄ClNO₂

Formula Weight: 287.75

CAS Number: 472981-92-3

Purity: >98%

Formulation: powder

Solubility: Soluble in DMSO (up to 25 mg/ml).

Storage: -20°C

Stability: ≥ 1 year.

 

Applications

TRPV1 blocker

 

Functions

SB-366791 is a potent (IC50 = 0.7 µM) and selective TRPV1 antagonist.  Selective for TRPV1 in a panel of 47 different binding assays.

 

Application Procedures

First dissolved in DMSO (up to 25 mg/ml), then diluted to aqueous buffer. Solutions in DMSO may be stored at -20°C for up to 3 months.

 

Additional information

SIZE (mg)	10 MG, 50 MG

TBI1217_SB-366791