Pyrilamine maleate (Mepyramine), Histamine receptor H1 inverse agonist; Sequesters G(q/11) (TBI3108)
$99.00 – $396.00
Histamine receptor H1 inverse agonist; Sequesters G(q/11)
| SKU | Stock | SIZE (mg) | Price | Quantity | ||
|---|---|---|---|---|---|---|
| TBI3108-5MG | Yes | 5 MG | $99.00 | |||
| TBI3108-25MG | Yes | 25 MG | $396.00 |
- Description
- Terms
- Additional information
- Documents
- Reviews (0)
Description
Product Details
Formal Name: (S)-α-Cyano-3-phenoxybenzyl (1R, 3R)-3-(2,2-dibromovinyl)-2,2-dimethylcyclopropanecarboxylate
Molecular Formula: C22H19Br2NO3
Formula Weight: 505.20
CAS Number: 59-33-6
Purity: >98%
Formulation: powder
Solubility: Soluble in DSMO (up to 50 mg/ml)
Storage: -20°C
Stability: ≥ 1 year.
Applications
Histamine receptor H1 inverse agonist; Sequesters G(q/11)
Functions
Reported to be an inhibitor of calcineurin (PP2B), IC50~100 pM but this activity has been disputed. Markedly enhances the expression of BDNF in cultured rat cortical neurons and displays neurotrophic effects. Produces antidepressant-like effects in mice. Blocks the spontaneous down-regulation of Nav1.8 sodium channels expressed in Xenopus oocytes.
Application Procedures
First dissolved in DSMO (up to 50 mg/ml), then diluted to aqueous buffer.
Research use only.
Additional information
| SIZE (mg) | 25 MG, 5 MG |
|---|
TBI3108_Pyrilamine_maleate(Mepyramine)
Research use only.
Be the first to review “Pyrilamine maleate (Mepyramine), Histamine receptor H1 inverse agonist; Sequesters G(q/11) (TBI3108)”
You must be logged in to post a review.
Reviews
There are no reviews yet.