MRL-24, PPARg partial agonist (TBI1365)
$117.00 – $468.00
PPARg partial agonist
SKU | Stock | SIZE (mg) | Price | Quantity | ||
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TBI1365-5MG | Yes | 5 MG | $117.00 | |||
TBI1365-25MG | Yes | 25 MG | $468.00 |
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Description
Product Details
Formal Name: (S)-2-(3-((1-(4-Methoxybenzoyl)-2-methyl-5-(trifluoromethoxy)-1H-indol-3-yl)methyl)phenoxy)propanoic acid
Molecular Formula: C28H24F3NO6
Formula Weight: 527.49
CAS Number: N/A
Purity: >98%
Formulation: powder
Solubility: Soluble in DMSO (up to 30 mg/ml)
Storage: -20°C
Stability: ≥ 2 years.
Applications
PPARg partial agonist
Functions
Displays high affinity for PPARγ with excellent anti-diabetic activity in mice but poor PPARγ agonist activity in transcription and adipogenesis assays. Highly effective (30 nM) at blocking Cdk5-mediated phosphorylation of PPARγ. Cell permeable.
Application Procedures
First dissolved in DMSO (up to 30 mg/ml), then diluted to aqueous buffer. Solutions in DMSO may be stored at -20°C for up to 2 months.
Additional information
SIZE (mg) | 25 MG, 5 MG |
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