CPTH2, HAT inhibitor (TBI4528)
$124.00 – $450.00
HAT inhibitor
SKU | Stock | SIZE (mg) | Price | Quantity | ||
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TBI4528-5MG | Yes | 5 MG | $124.00 | |||
TBI4528-25MG | Yes | 25 MG | $450.00 |
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Description
Product Details
Formal Name: Cyclopentylidene-[4-(4’-chlorophenyl)thiazol-2-yl]hydrazone
Molecular Formula: C14H14ClN3S
Formula Weight: 291.80
CAS Number: 357649-93-5
Purity: >98%
Formulation: powder
Solubility: Soluble in DMSO (up to 25 mg/ml).
Storage: -20°C
Stability: ≥ 1 year.
Applications
HAT inhibitor
Functions
CPTH2 is a selective inhibitor of the histone acetyltransferase Gcn5P both in vitro and in vivo (IC50 = 0.80 mM). In vitro, the HAT inhibitory activity of CPTH2 was caused via bridge-interaction with histone H3. In vivo it decreased acetylation of bulk histone H3 at the H3-AcK14 site.
Application Procedures
First dissolved in DMSO (up to 25 mg/ml), then diluted to aqueous buffer. Solutions in DMSO may be stored at -20° for up to 1 month.
Additional information
SIZE (mg) | 25 MG, 5 MG |
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