MK-571, Leukotriene Cys LT1 antagonist (TBI1039)
$108.00 – $432.00
Leukotriene Cys LT1 antagonist
SKU | Stock | SIZE (mg) | Price | Quantity | ||
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TBI1039-5MG | Yes | 5 MG | $108.00 | |||
TBI1039-25MG | Yes | 25 MG | $432.00 |
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Description
Product Details
Formal Name: 5-(3-(2-(7-Chloroquinolin-2-yl)ethenyl)phenyl)-8-dimethylcarbamyl-4,6-dithiaoctanoic acid, sodium salt
Alternate Names: L-660711
Molecular Formula: C26H26ClN2O3S2 · Na
Formula Weight: 537.10
CAS Number: 115104-28-4
Purity: >98%
Formulation: powder
Solubility: Soluble in DMSO (up to 50 mg/ml).
Storage: RT
Stability: ≥ 1 year.
Applications
Leukotriene Cys LT1 antagonist
Functions
Potent (EC50 = 1.3nM) and selective Leukotriene D4 antagonist(LTD4) displaying inverse agonist activity, Blocks binding of LTD4 to human (Ki = 0.22 nM) and guinea pig (Ki = 2.1 nM) lung membranes. Selective for the CysLT1 receptor. Multidrug resistance protein 1 (MRP1) inhibitor.
Application Procedures
First dissolved in DMSO (up to 50 mg/ml), then diluted to aqueous buffer. Solutions in DMSO may be stored at -20°C for up to 2 months.
Additional information
SIZE (mg) | 25 MG, 5 MG |
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