C-646, HAT inhibitor (TBI1306)
$144.00 – $576.00
HAT inhibitor
SKU | Stock | SIZE (mg) | Price | Quantity | ||
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TBI1306-5MG | Yes | 5 MG | $144.00 | |||
TBI1306-25MG | Yes | 25 MG | $576.00 |
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Description
Product Details
Formal Name: 4-[4-[[5-(4,5-Dimethyl-2-nitrophenyl)-2-furanyl]methylene]-4,5-dihydro-3-methyl-5-oxo-1H-pyrazol-1-yl]benzoic acid
Molecular Formula: C24H19N3O6
Formula Weight: 445.44
CAS Number: 328968-36-1
Purity: >98%
Formulation: powder
Solubility: Soluble in DMSO (up to 10 mg/ml).
Storage: -20°C
Stability: ≥ 2 years.
Applications
HAT inhibitor
Functions
Potent and selective inhibitor of the histone acetyl transferase p300/CBP (Ki=400 nM ). Induces apoptosis in prostate cancer cells. Enhances fear extinction memory and synaptic plasticity in mice. Promotes tau deacetylation reducing levels of pathogenic p-tau. Cell permeable.
Application Procedures
First dissolved in DMSO (up to 10 mg/ml), then diluted to aqueous buffer. Solutions in DMSO may be stored at -20° for up to 2 months.
Additional information
SIZE (mg) | 25 MG, 5 MG |
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