AH-7614, GPR120 antagonist (TBI1521)
$81.00 – $324.00
GPR120 antagonist
SKU | Stock | SIZE (mg) | Price | Quantity | ||
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TBI1521-5MG | Yes | 5 MG | $81.00 | |||
TBI1521-25MG | Yes | 25 MG | $324.00 |
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Description
Product Details
Formal Name: 4-Methyl-N-9H-xanthen-9-yl-benzenesulfonamide
Molecular Formula: C20H17NO3S
Formula Weight: 351.43
CAS Number: 6326-06-3
Purity: >98%
Formulation: powder
Solubility: Soluble in DMSO (up to 50 mg/ml) or in Ethanol (up to 8 mg/ml with warming).
Storage: -20°C
Stability: ≥ 2 years.
Applications
GPR120 antagonist
Functions
Selective antagonist at free fatty acid receptor 4 (FFA4), also known as GPR120. pIC50s= 7.1 and <4.6 for FFA4 and FFA1 respectively. Inhibits linoleic acid and GSK137647A-induced intracellular calcium increase in U2OS osteosarcoma cells expressing GPR120. Has been used to probe the GPR120-mediated effects of fatty acids on a GnRH-synthesizing neuronal cell model.
Application Procedures
First dissolved in DMSO (up to 50 mg/ml) or in Ethanol (up to 8 mg/ml with warming), then diluted to aqueous buffer. Solutions in DMSO or ethanol may be stored at -20° for up to 1 month.
Additional information
SIZE (mg) | 25 MG, 5 MG |
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