NADA, Endogenous TRPV1 activator (TBI1479)
$83.00 – $328.00
Endogenous TRPV1 activator
SKU | Stock | SIZE (mg) | Price | Quantity | ||
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TBI1479-5MG | Yes | 5 MG | $83.00 | |||
TBI1479-25MG | Yes | 25 MG | $328.00 |
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Description
Product Details
Formal Name: N-(5Z,8Z,11Z,14Z-eicosatetraenoyl)dopamine
Alternate Names: NADA; AA-DA; N-Arachidonoyldopamine
Molecular Formula: C28H41NO3
Formula Weight: 439.63
CAS Number: 199875-69-9
Purity: >98%
Formulation: oil
Solubility: Soluble in DMSO (up to 50 mg/ml)
Storage: -20°C
Stability: ≥ 2 years.
Applications
Endogenous TRPV1 activator
Functions
Endogenous conjugate of arachidonic acid and dopamine. May be the “endogenous capsaicin like substance” in the CNS acting at TRPV1 channels, EC50~ 50 nM1. Also acts as a selective cannabinoid CB1 agonist (Ki=0.25 and 15 μM for CB1 and CB2 respectively) and results in a distinct signaling profile from any known cannabinoid. Competitive inhibitor of FAAH and anadamide transport. Modulates acute systemic inflammation via non-hematopoietic TRPV1.
Application Procedures
First dissolved in DMSO (up to 50 mg/ml), then diluted to aqueous buffer. Subject to air oxidation Solutions in DMSO may be stored at -80° under an inert atmosphere for up to 1 month.
Additional information
SIZE (mg) | 25 MG, 5 MG |
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