BI-9564, BRD9 bromodomain inhibitor (TBI4320)
$108.00 – $351.00
BRD9 bromodomain inhibitor
SKU | Stock | SIZE (mg) | Price | Quantity | ||
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TBI4320-5MG | Yes | 5 MG | $108.00 | |||
TBI4320-25MG | Yes | 25 MG | $351.00 |
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Description
Product Details
Formal Name: 4-[4-[(Dimethylamino)methyl]-2,5-dimethoxyphenyl]-2-methyl-2,7-naphthyridine-1-one
Molecular Formula: C20H23N3O3
Formula Weight: 353.40
CAS Number: 1883429-22-8
Purity: >98%
Formulation: powder
Solubility: Soluble in DMSO (up to 5 mg/ml)
Storage: -20°C
Stability: ≥ 2 years.
Applications
BRD9 bromodomain inhibitor
Functions
Potent, selective, and cell permeable inhibitor of the BRD9 bromodomain, a subunit of the switch/sucrose nonfermentable (SWI/SNF) chromatin remodeling complex (IC50 = 75 nM). It displayed antitumor activity in an acute myeloid leukemia xenograft model. BI-9564 displayed cytotoxic and anti-proliferative effects in 5 rhabdoid tumor cell lines.
Application Procedures
First dissolved in DMSO (up to 5 mg/ml), then diluted to aqueous buffer. Solutions in DMSO may be stored at -20°C for up to 3 months.
Additional information
SIZE (mg) | 25 MG, 5 MG |
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