PSB-CB5, GPR18 antagonist (TBI5062)
$135.00 – $540.00
GPR18 antagonist
SKU | Stock | SIZE (mg) | Price | Quantity | ||
---|---|---|---|---|---|---|
TBI5062-5MG | Yes | 5 MG | $135.00 | |||
TBI5062-25MG | Yes | 25 MG | $540.00 |
- Description
- Terms
- Additional information
- Documents
- Reviews (0)
Description
Product Details
Formal Name: (2Z)-2[[3-[(4-Chlorophenyl)methoxy]phenyl]methylene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3(2H)-one
Alternate Names: CID-85469571
Molecular Formula: C20H17ClN2O2S
Formula Weight: 384.88
CAS Number: 1627710-30-8
Purity: >98%
Formulation: powder
Solubility: Soluble in DMSO (up to 25 mg/ml)
Storage: -20°C
Stability: ≥ 1 year.
Applications
GPR18 antagonist
Functions
A potent and selective GPR18 antagonist (IC50 = 0.279 µM) exhibiting >36-fold selectivity against GPR55 and CB1 and 14-fold selectivity against CB2. Inhibits N-arachidonylglycine-induced acrosomal exocytosis in human spermatozoa indicating that GPR18 may be involved in physiological processes of human spermatozoa.
Application Procedures
First dissolved in DMSO (up to 25 mg/ml), then diluted to aqueous buffer. Solutions in DMSO may be stored at -20°C for up to 3 months.
Additional information
SIZE (mg) | 25 MG, 5 MG |
---|
Be the first to review “PSB-CB5, GPR18 antagonist (TBI5062)”
You must be logged in to post a review.
Reviews
There are no reviews yet.