Palmitoylethanolamide, GPR55 agonist; endogenous cannabinoid (TBI1297)

Description

Product Details

Formal Name: N-(2-hydroxyethyl)palmitamide

Alternate Names: PEA

Molecular Formula: C₁₈H₃₇NO₂

Formula Weight: 299.50

CAS Number: 544-31-0

Purity: >98%

Formulation: powder

Solubility: Soluble in DMSO (up to 25 mg/ml) or in Ethanol (up to 25 mg/ml).

Storage: -20°C

Stability: ≥ 2 years.

 

Applications

GPR55 agonist; endogenous cannabinoid

 

Functions

Endogenous cannabinoid. Weak ligand for CB1 (Ki=23.8 µM) and CB2 (Ki=13.9 µM) receptor.  Selective agonist at GPR55. Inhibits expression of fatty acid amide hydrolase (FAAH). Displays immunosuppressant and anti-inflammatory activity and reduces granuloma-induced hyperalgesia.

 

Application Procedures

First dissolved in DMSO (up to 25 mg/ml) or in Ethanol (up to 25 mg/ml), then diluted to aqueous buffer. Solutions in water may be stored at -20°C for up to 3 months.

Additional information

SIZE (mg)	20 MG, 100 MG

TBI1297_Palmitoylethanolamide