KT-5823, PKG inhibitor (TBI2083)
$175.00 – $700.00
SKU | Stock | SIZE | Price | Quantity | ||
---|---|---|---|---|---|---|
TBI2083-100UG | Yes | 100 µg | $175.00 | |||
TBI2083-500UG | Yes | 500 µg | $700.00 |
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Description
Product Details
Molecular Formula: C29H25N3O5
Formula Weight: 495.50
CAS Number: 126643-37-6
Purity: >98%
Formulation: Powder
Solubility: Soluble in DMSO (up to 25 mg/ml) or in DMF (up to 20 mg/ml).
Storage: -20°C
Stability: ≥ 2 years.
Applications
- PKG inhibitor
Functions
KT5823 (126643-37-6) is a selective protein kinase G inhibitor (K>i =0.23, 4 and >10 μM for PKG, PKC and PKA respectively. Arrests human skin fibroblast cell cycle after the G0/G1 boundary. KT5823 abolishes the cGMP-induced relaxation in smooth muscle cells (IC50=60 nM). Cell permeable.
Application Procedures
First dissolved in DMSO (up to 25 mg/ml) or in DMF (up to 20 mg/ml), then diluted to aqueous buffer. Solutions in DMSO or DMF may be stored at -20°C for up to 3 months.
Additional information
SIZE | 100 µg, 500 µg |
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