GRI-977143, LPA2 antagonist (TBI1442)
$144.00 – $576.00
LPA2 antagonist
SKU | Stock | SIZE (mg) | Price | Quantity | ||
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TBI1442-5MG | Yes | 5 MG | $144.00 | |||
TBI1442-25MG | Yes | 25 MG | $576.00 |
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Description
Product Details
Formal Name: 2-[[3-(1,3-dioxo-1H-benz[de]isoquinolin-2(3H)-yl)propyl]thio]benzoic acid
Molecular Formula: C22H17NO6S
Formula Weight: 391.44
CAS Number: 325850-81-5
Purity: >98%
Formulation: powder
Solubility: Soluble in DMSO (up to 35 mg/ml)
Storage: -20°C
Stability: ≥ 1 year.
Applications
LPA2 antagonist
Functions
Selective agonist of the lysophosphatidic acid – 2 (LPA2) receptor. Displays antiapoptotic activity. Rescues apoptotically condemned cells from death and injury caused by high-dose γ-irradiation in vitro and in vivo. Rescues mice from deadly levels of radiation when given 24 hours post-exposure. Activates the ERK1/2 prosurvival pathway.
Application Procedures
First dissolved in DMSO (up to 35 mg/ml), then diluted to aqueous buffer. Solutions in DMSO may be stored at -20°C for up to 3 months.
Additional information
SIZE (mg) | 25 MG, 5 MG |
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