GDC-0941, pan-PI3K inhibitor (TBI2141)
$104.00 – $288.00
pan-PI3K inhibitor
SKU | Stock | SIZE (mg) | Price | Quantity | ||
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TBI2141-5MG | Yes | 5 MG | $104.00 | |||
TBI2141-25MG | Yes | 25 MG | $288.00 |
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Description
Product Details
Alternate Names: Pictilisib
Molecular Formula: C23H27N7O3S2
Formula Weight: 513.64
CAS Number: 957054-30-7
Purity: >98%
Formulation: powder
Solubility: Soluble in DMSO (up to 50 mg/ml).
Storage: -20°C
Stability: ≥ 1 year.
Applications
pan-PI3K inhibitor
Functions
GDC-0941 is a potent and selective inhibitor of class I phosphatidylinositol-3-kinases (PI3K) with significant antitumor activity – IC50’s: PI3Kα = 3nM, PI3Kβ = 33 nM, PI3Kδ = 3 nM, PI3Kγ = 75 nM. GDC-0941 is the chemical probe of choice for the pan-inhibition of class I PI3K’s. Currently in clinical trials.
Application Procedures
First dissolved in DMSO (up to 50 mg/ml), then diluted to aqueous buffer. Solutions in DMSO may be stored at -20°C for up to 3 months.
Additional information
SIZE (mg) | 25 MG, 5 MG |
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