Calphostin C, Protein Kinase C inhibitor (TBI5635)
$263.00 – $1,206.00
Protein Kinase C inhibitor
SKU | Stock | SIZE | Price | Quantity | ||
---|---|---|---|---|---|---|
TBI5635-100UG | Yes | 100 µg | $263.00 | |||
TBI5635-500UG | Yes | 500 µg | $1,206.00 |
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Description
Product Details
Formal Name: Fermentation product from Cladisporium cladosporioides
Alternate Names: UCN-1028C; PKF115-584
Molecular Formula: C44H38O14
Formula Weight: 790.80
CAS Number: 121263-19-2
Purity: >95%
Formulation: powder
Solubility: Soluble in DMSO (10 mg/ml)
Storage: -20°C
Stability: ≥ 1 year.
Applications
Protein Kinase C inhibitor
Functions
A potent and specific inhibitor of protein kinase C (PKC, IC50 = 50 nM). Inhibition of PKC is light dependent and is competitive with the diacylglycerol / phorbol ester binding site. Calphostin C competes with the diacylglycerol / phorbol ester binding site in other proteins such as Munc13-1. Reverses oxycodone-induced tolerance to respiratory depression.
Application Procedures
First dissolved in DMSO (10 mg/ml), then diluted to aqueous buffer. Solutions in DMSO may be stored at -20°C for up to 3 months.
Additional information
SIZE | 100 µg, 500 µg |
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