RGFP966, Selective HDAC3 inhibitor (TBI4029)
$126.00 – $486.00
Selective HDAC3 inhibitor
SKU | Stock | SIZE (mg) | Price | Quantity | ||
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TBI4029-5MG | Yes | 5 MG | $126.00 | |||
TBI4029-25MG | Yes | 25 MG | $486.00 |
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Description
Product Details
Formal Name: (2E)-N-(2-Amino-4-fluorophenyl)-3-[(2E)-1-(3-phenyl-2-propen-1-yl)-1H-pyrazol-4-yl]-2-propenamide
Molecular Formula: C21H19FN4O
Formula Weight: 362.40
CAS Number: 1357389-11-7
Purity: >98%
Formulation: powder
Solubility: Soluble in DMSO (up to 20 mg/ml)
Storage: -20°C
Stability: ≥ 1 year.
Applications
Selective HDAC3 inhibitor
Functions
RGFP966 is a selective inhibitor of HDAC3 (IC50 = 80 nM, no other HDACs inhibited at 15µM). It facilitates the extinction of cocaine-seeking behavior in mice and transforms subthreshold learning events into robust long-term memory, suggesting a potential therapeutic target for memory enhancement and neurodegenerative diseases.
Application Procedures
First dissolved in DMSO (up to 20 mg/ml), then diluted to aqueous buffer. Solutions in DMSO may be stored at -20°C for up to 1 month.
Additional information
SIZE (mg) | 25 MG, 5 MG |
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