SKF-525A HCl, Cytochrome P450 inhibitor (TBI4050)
$90.00 – $369.00
Cytochrome P450 inhibitor
SKU | Stock | SIZE (mg) | Price | Quantity | ||
---|---|---|---|---|---|---|
TBI4050-100MG | Yes | 100 MG | $90.00 | |||
TBI4050-500MG | Yes | 500 MG | $369.00 |
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Description
Product Details
Formal Name: N,N-Diethylaminoethyl-2,2-diphenylvalerate hydrochloride
Alternate Names: Proadifen
Molecular Formula: C23H31NO2 ∙ HCl
Formula Weight: 390.00
CAS Number: 62-68-0
Purity: >98%
Formulation: powder
Solubility: Soluble in DMSO (up to 20 mg/ml)
Storage: -20°C
Stability: ≥ 1 year.
Applications
Cytochrome P450 inhibitor
Functions
Broad-spectrum cytochrome P450 monoxygenase inhibitor that also blocks the acetylcholine receptor (IC50 = 19 µM). Inhibits nitric oxide synthase (NOS). Also inhibits glibenclamide-sensitive K+ channels (IC50 = 9.8 µM) in Xenopus oocytes. Increases inflammatory cytokine expression in Müller glial cells and inhibits the excitability of rat 5-HT neurons.
Application Procedures
First dissolved in DMSO (up to 20 mg/ml), then diluted to aqueous buffer. Solutions in DMSO may be stored at -20°C for up to 3 months.
Additional information
SIZE (mg) | 500 MG, 100 MG |
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