A-803467, Sodium NaV1.8 channel blocker (TBI1066)
$90.00 – $360.00
Sodium NaV1.8 channel blocker
SKU | Stock | SIZE (mg) | Price | Quantity | ||
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TBI1066-10MG | Yes | 10 MG | $90.00 | |||
TBI1066-50MG | Yes | 50 MG | $360.00 |
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Description
Product Details
Formal Name: 5-(4-Chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-carboxamide
Molecular Formula: C19H16ClNO4
Formula Weight: 357.80
CAS Number: 944361-79-4
Purity: >98%
Formulation: powder
Solubility: Soluble in DMSO (up to 15 mg/ml) or in Ethanol (up to 2 mg/ml).
Storage: RT
Stability: ≥ 1 year.
Applications
Sodium NaV1.8 channel blocker
Functions
Potent, selective inhibitor of the TTX-resistant voltage-gated sodium channel Nav1.8. Nav1.8 is preferentially expressed in sensory neurons, and inhibition attenuates both inflammatory and neuropathic pain in a variety of animal models. IC50’s for rat and human Nav1.8 are 140 nM and 8.0 nM respectively.
Application Procedures
First dissolved in DMSO (up to 15 mg/ml) or in Ethanol (up to 2 mg/ml), then diluted to aqueous buffer. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.
Additional information
SIZE (mg) | 10 MG, 50 MG |
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