H89 · 2HCl, PKA inhibitor (TBI2144)
$90.00 – $324.00
PKA inhibitor
SKU | Stock | SIZE (mg) | Price | Quantity | ||
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TBI2144-5MG | Yes | 5 MG | $90.00 | |||
TBI2144-25MG | Yes | 25 MG | $324.00 |
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Description
Product Details
Formal Name: N-[2-[[3-(4-Bromophenyl)-2-propen-1-yl]amino]ethyl]-5-isoquinolinesulfonamide dihydrochloride
Molecular Formula: C20H20BrN3O2S·2HCl
Formula Weight: 519.28
CAS Number: 127243-85-0
Purity: >98%
Formulation: Powder
Solubility: Soluble in DMSO (up to 50 mg/ml) or in Water (up to 10 mg/ml).
Storage: -20°C
Stability: ≥ 2 years.
Applications
- PKA inhibitor
Functions
H-89 (127243-85-0) is a commonly used inhibitor of protein kinase A (PKA IC50 = 140 nM). Inhibits a variety of other kinases including S6K1 (IC50 = 80 nM), MSK1 (120 nM), ROCK II (270 nM), PKBα (2.6 µM), PKD, PRK2, RSK1 and 2, SGK, AMPK, CHK1 and MAPKAP-K1b (2.8 µM).
Application Procedures
Solutions in DMSO or distilled water may be stored at -20°C for up to 3 months.
Additional information
SIZE (mg) | 25 MG, 5 MG |
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